China (Mainland)
Best price 4093-35-0 in stock Bromopride manufacturer CAS NO.4093-35-0
- Min.Order: 0 Metric Ton
- Payment Terms: L/C,D/A,D/P,T/T,
- Product Details
Keywords
- Best price 4093-35-0
- Bromopride 4093-35-0 in stock
- Bromopride manufacturer
Quick Details
- ProName: Best price 4093-35-0 in stock Bromopri...
- CasNo: 4093-35-0
- Molecular Formula: C14H22 Br N3 O2
- DeliveryTime: one week
- Port: shanghai
- ProductionCapacity: 5-10 Metric Ton/Year
- Purity: 99%
- Storage: 500kg in stock
- LimitNum: 0 Metric Ton
Superiority
Bromopride is a dopamine D2 receptor antagonist (Ki = 14 nM).It binds to bovine anterior pituitary membranes with an IC50 value of 2.13 μM. Bromopride inhibits cholinesterase activity in vitro in rat plasma and striatum homogenate (IC50s = 67.8 and 38.4 μM, respectively). It increases serum prolactin levels in rats by 100% when used at a dose of 0.02 mol/kg. Bromopride (2.5 mg/kg) decreases locomotion and rearing in an open field test and impairs acquistion, but not retention, of a conditioned avoidance response in a two-way active conditioned avoidance test in rats.
Bromopride (free base) is a dopamine antagonist with prokinetic properties widely used as an antiemetic
Details
Bromopride is a dopamine antagonist used as an antiemetic. Its prokinetic properties are similar to those of metoclopramide. It is unavailable in America or the United Kingdom.
Bromopride is a dopamine antagonist with prokinetic properties, widely used as an antiemetic.
| Catalogue Number | B686645 |
| Chemical Name | Bromopride |
| Synonyms | 4-Amino-5-bromo-N-[2-(diethylamino)ethyl]-2-methoxybenzamide; 2-Methoxy-4-amino-5-bromo-N,N-diethylaminoethylbenzamide; N-Diethylaminoethyl-2-methoxy-4-amino-5-bromobenzamide; Emepride; Emoril; Viadil |
| CAS Number | 4093-35-0 |
| Molecular Formula | C??H??BrN?O? |
| Appearance | White to Off-White Solid |
| Melting Point | 148 - 150°C |
| Molecular Weight | 344.25 |
| Storage | Refrigerator |
| Solubility | Chloroform (Slightly), DMSO (Slightly), Methanol (Slightly) |
| Category | Standards; Pharmaceutical/API Drug Impurities/Metabolites; |
| Applications | An antiemetic. Bromopride is used in method and a system for analyzing neuropharmacology of a drug. |